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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50202959'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM50202959
PNG
((+/-)-1-[2-(4-fluorophenyl)-2-(4-methylpiperazin-1...)
Show SMILES CN1CCN(CC1)C(CN1CCN(CCCCCc2cccc3ccccc23)CC1)c1ccc(F)cc1 |w:7.8|
Show InChI InChI=1S/C32H43FN4/c1-34-18-24-37(25-19-34)32(29-13-15-30(33)16-14-29)26-36-22-20-35(21-23-36)17-6-2-3-8-27-10-7-11-28-9-4-5-12-31(27)28/h4-5,7,9-16,32H,2-3,6,8,17-26H2,1H3
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Similars
Article
PubMed
n/an/a 218n/an/an/an/an/an/a



Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL


Assay Description
Displacement of [125I]Nle4-D-Phe7-alpha-MSH from human MC4 receptor expressed in COS1 cells

Bioorg Med Chem 15: 1989-2005 (2007)


Article DOI: 10.1016/j.bmc.2006.12.039
BindingDB Entry DOI: 10.7270/Q2C53KHN
More data for this
Ligand-Target Pair