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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50202965'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM50202965
PNG
((+/-)-1-(1-(4-fluorophenyl)-2-{4-[4-(4-methoxy-1-n...)
Show SMILES COc1ccc(CCCCN2CCN(CC(N3CCN(C)CC3)c3ccc(F)cc3)CC2)c2ccccc12 |w:15.14|
Show InChI InChI=1S/C32H43FN4O/c1-34-17-23-37(24-18-34)31(27-10-13-28(33)14-11-27)25-36-21-19-35(20-22-36)16-6-5-7-26-12-15-32(38-2)30-9-4-3-8-29(26)30/h3-4,8-15,31H,5-7,16-25H2,1-2H3
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Similars
Article
PubMed
n/an/a 228n/an/an/an/an/an/a



Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL


Assay Description
Displacement of [125I]Nle4-D-Phe7-alpha-MSH from human MC4 receptor expressed in COS1 cells

Bioorg Med Chem 15: 1989-2005 (2007)


Article DOI: 10.1016/j.bmc.2006.12.039
BindingDB Entry DOI: 10.7270/Q2C53KHN
More data for this
Ligand-Target Pair