Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 1 (RAT) | BDBM50098248 (2-Amino-3-(3-hydroxy-4-phenyl-isoxazol-5-yl)-propi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description The compound was tested for the receptor binding affinity at Metabotropic glutamate receptor 1 using established second messenger assay systems. | J Med Chem 45: 988-91 (2002) BindingDB Entry DOI: 10.7270/Q2M32V27 | |||||||||||
More data for this Ligand-Target Pair |