Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 8 (Rattus norvegicus (Rat)) | BDBM82006![]() (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Toronto Curated by PDSP Ki Database | Neuropharmacology 40: 170-7 (2001) Article DOI: 10.1016/s0028-3908(00)00128-3 BindingDB Entry DOI: 10.7270/Q27P8WZ1 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 8 (Rattus norvegicus (Rat)) | BDBM82006![]() (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 290 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair |