BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase' and Ligand = 'BDBM50169678'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Methionine aminopeptidase


(Escherichia coli (strain K12))
BDBM50169678
PNG
(5-(3-Chloro-benzoylamino)-thiazole-4-carboxylic ac...)
Show SMILES Clc1cccc(c1)C(=O)Nc1scnc1C(=O)Nc1nccs1
Show InChI InChI=1S/C14H9ClN4O2S2/c15-9-3-1-2-8(6-9)11(20)18-13-10(17-7-23-13)12(21)19-14-16-4-5-22-14/h1-7H,(H,18,20)(H,16,19,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 270n/an/an/an/an/an/a



Graduate School of the Chinese Academy of Sciences

Curated by ChEMBL


Assay Description
Inhibitory concentration required against Escherichia coli MetAP1 (150 nM)


Bioorg Med Chem Lett 15: 3732-6 (2005)


Article DOI: 10.1016/j.bmcl.2005.05.055
BindingDB Entry DOI: 10.7270/Q2T1534B
More data for this
Ligand-Target Pair