BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase' and Ligand = 'BDBM50169685'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Methionine aminopeptidase


(Escherichia coli (strain K12))
BDBM50169685
PNG
(CHEMBL360353 | N-[4-(Thiazol-2-ylcarbamoyl)-thiazo...)
Show SMILES CCOC(=O)CC(=O)Nc1scnc1C(=O)Nc1nccs1
Show InChI InChI=1S/C12H12N4O4S2/c1-2-20-8(18)5-7(17)15-11-9(14-6-22-11)10(19)16-12-13-3-4-21-12/h3-4,6H,2,5H2,1H3,(H,15,17)(H,13,16,19)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 66n/an/an/an/an/an/a



Graduate School of the Chinese Academy of Sciences

Curated by ChEMBL


Assay Description
Inhibitory concentration required against Escherichia coli MetAP1 (150 nM)


Bioorg Med Chem Lett 15: 3732-6 (2005)


Article DOI: 10.1016/j.bmcl.2005.05.055
BindingDB Entry DOI: 10.7270/Q2T1534B
More data for this
Ligand-Target Pair