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Found 1 hit Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase' and Ligand = 'BDBM50497537'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Methionine aminopeptidase


(Escherichia coli (strain K12))		BDBM50497537
PNG
(CHEMBL3337628)
Show SMILES Cl.COc1ccc2CCC(CN3CCCCC3)C(=O)c2c1
Show InChI InChI=1S/C17H23NO2.ClH/c1-20-15-8-7-13-5-6-14(17(19)16(13)11-15)12-18-9-3-2-4-10-18;/h7-8,11,14H,2-6,9-10,12H2,1H3;1H
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 3.70E+3n/an/an/an/an/an/a



Heidelberg University

Curated by ChEMBL


Assay Description
Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...

Bioorg Med Chem Lett 24: 5310-4 (2014)


Article DOI: 10.1016/j.bmcl.2014.09.047
BindingDB Entry DOI: 10.7270/Q2057JW8
More data for this
Ligand-Target Pair