Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase 2' and Ligand = 'BDBM188711'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM188711 (US9169246, 253) Show SMILES FC(F)(F)Cn1c2cc(ccc2c2[nH]ncc2c1=O)-c1cccnc1N1CCNC(=O)C1 Show InChI InChI=1S/C21H17F3N6O2/c22-21(23,24)11-30-16-8-12(3-4-14(16)18-15(20(30)32)9-27-28-18)13-2-1-5-26-19(13)29-7-6-25-17(31)10-29/h1-5,8-9H,6-7,10-11H2,(H,25,31)(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	9.44	n/a	n/a	n/a	n/a	n/a	n/a
SANOFI US Patent					Assay Description The enzymatic test is a test in two steps.In a first step, it consists in placing in contact the compound according to the invention, the dialysed Me...				US Patent US9169246 (2015) BindingDB Entry DOI: 10.7270/Q2B856XZ
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