Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Monoglyceride lipase (Homo sapiens (Human)) | BDBM50049459 (CHEMBL3318314) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Jamia Hamdard (Hamdard University) Curated by ChEMBL | Assay Description Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 mins | Bioorg Med Chem Lett 24: 3986-96 (2014) Article DOI: 10.1016/j.bmcl.2014.06.029 BindingDB Entry DOI: 10.7270/Q2XP76J6 | |||||||||||
More data for this Ligand-Target Pair |