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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mucosa-associated lymphoid tissue lymphoma translocation protein 1' and Ligand = 'BDBM487669'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mucosa-associated lymphoid tissue lymphoma translocation protein 1


(Homo sapiens (Human))		BDBM487669
PNG
(N-(5-chloro-6-(oxazol-2- yl)pyridin-3-yl)-1-(quino...)
Show SMILES FC(F)(F)c1c(cnn1-c1cccc2ncccc12)C(=O)Nc1cnc(-c2ncco2)c(Cl)c1
Show InChI InChI=1S/C22H12ClF3N6O2/c23-15-9-12(10-29-18(15)21-28-7-8-34-21)31-20(33)14-11-30-32(19(14)22(24,25)26)17-5-1-4-16-13(17)3-2-6-27-16/h1-11H,(H,31,33)
PDB

UniProtKB/SwissProt

GoogleScholar
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PC cid
PC sid
UniChem
US Patent
n/an/a 15n/an/an/an/an/an/a



Janssen Pharmaceutica NV

US Patent


Assay Description
MALT1 protease activity was assessed in an in vitro assay using a tetrapeptide as substrate and full-length MALT1 protein (Strep-MALT1(1-824)-His) pu...

US Patent US10954214 (2021)


BindingDB Entry DOI: 10.7270/Q2SX6HB1
More data for this
Ligand-Target Pair