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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mucosa-associated lymphoid tissue lymphoma translocation protein 1' and Ligand = 'BDBM487704'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mucosa-associated lymphoid tissue lymphoma translocation protein 1


(Homo sapiens (Human))		BDBM487704
PNG
(N-(5-cyano-6-(2H-1,2,3-triazol- 2-yl)pyridin-3-yl)...)
Show SMILES FC(F)(F)c1c(cnn1-c1ccnc2sccc12)C(=O)Nc1cnc(c(c1)C#N)-n1nccn1
Show InChI InChI=1S/C20H10F3N9OS/c21-20(22,23)16-14(10-29-31(16)15-1-3-25-19-13(15)2-6-34-19)18(33)30-12-7-11(8-24)17(26-9-12)32-27-4-5-28-32/h1-7,9-10H,(H,30,33)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 15n/an/an/an/an/an/a



Janssen Pharmaceutica NV

US Patent


Assay Description
MALT1 protease activity was assessed in an in vitro assay using a tetrapeptide as substrate and full-length MALT1 protein (Strep-MALT1(1-824)-His) pu...

US Patent US10954214 (2021)


BindingDB Entry DOI: 10.7270/Q2SX6HB1
More data for this
Ligand-Target Pair