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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mucosa-associated lymphoid tissue lymphoma translocation protein 1' and Ligand = 'BDBM487971'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mucosa-associated lymphoid tissue lymphoma translocation protein 1


(Homo sapiens (Human))		BDBM487971
PNG
(4-(4-((5-chloro-2-methyl-6-(2H- 1,2,3-triazol-2-yl...)
Show SMILES Cc1nc(c(Cl)cc1NC(=O)c1cnn(c1C(F)(F)F)-c1cnc(C(N)=O)c2sccc12)-n1nccn1
Show InChI InChI=1S/C21H13ClF3N9O2S/c1-9-13(6-12(22)19(31-9)34-28-3-4-29-34)32-20(36)11-7-30-33(17(11)21(23,24)25)14-8-27-15(18(26)35)16-10(14)2-5-37-16/h2-8H,1H3,(H2,26,35)(H,32,36)
PDB

UniProtKB/SwissProt

GoogleScholar
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PC cid
PC sid
UniChem
US Patent
n/an/a 12n/an/an/an/an/an/a



Janssen Pharmaceutica NV

US Patent


Assay Description
MALT1 protease activity was assessed in an in vitro assay using a tetrapeptide as substrate and full-length MALT1 protein (Strep-MALT1(1-824)-His) pu...

US Patent US10954214 (2021)


BindingDB Entry DOI: 10.7270/Q2SX6HB1
More data for this
Ligand-Target Pair