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Found 1 hit Enz. Inhib. hit(s) with Target = 'Mucosa-associated lymphoid tissue lymphoma translocation protein 1' and Ligand = 'BDBM50516114'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mucosa-associated lymphoid tissue lymphoma translocation protein 1


(Homo sapiens (Human))		BDBM50516114
PNG
(CHEMBL4536750)
Show SMILES COc1ccc(NC(=O)C2CCN(CC2)c2nccn3cccc23)cc1Cl
Show InChI InChI=1S/C20H21ClN4O2/c1-27-18-5-4-15(13-16(18)21)23-20(26)14-6-10-25(11-7-14)19-17-3-2-9-24(17)12-8-22-19/h2-5,8-9,12-14H,6-7,10-11H2,1H3,(H,23,26)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.10E+3n/an/an/an/an/an/a



Janssen Research & Development, LLC

Curated by ChEMBL


Assay Description
Inhibition of strep-tagged and His-tagged full length MALT1 protease (1 to 824 residues) (unknown origin) expressed in baculovirus infected insect ce...

Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126743
BindingDB Entry DOI: 10.7270/Q2DV1P7R
More data for this
Ligand-Target Pair