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Found 1 hit Enz. Inhib. hit(s) with Target = 'Mucosa-associated lymphoid tissue lymphoma translocation protein 1' and Ligand = 'BDBM50516139'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mucosa-associated lymphoid tissue lymphoma translocation protein 1


(Homo sapiens (Human))		BDBM50516139
PNG
(CHEMBL4565085)
Show SMILES Clc1cccnc1N1CCC(CC1)C(=O)Nc1cnc(Oc2cccnc2)c(Cl)c1
Show InChI InChI=1S/C21H19Cl2N5O2/c22-17-4-2-8-25-19(17)28-9-5-14(6-10-28)20(29)27-15-11-18(23)21(26-12-15)30-16-3-1-7-24-13-16/h1-4,7-8,11-14H,5-6,9-10H2,(H,27,29)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 130n/an/an/an/an/an/a



Janssen Research & Development, LLC

Curated by ChEMBL


Assay Description
Inhibition of strep-tagged and His-tagged full length MALT1 protease (1 to 824 residues) (unknown origin) expressed in baculovirus infected insect ce...

Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126743
BindingDB Entry DOI: 10.7270/Q2DV1P7R
More data for this
Ligand-Target Pair