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Found 1 hit Enz. Inhib. hit(s) with Target = 'Mucosa-associated lymphoid tissue lymphoma translocation protein 1' and Ligand = 'BDBM50516143'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mucosa-associated lymphoid tissue lymphoma translocation protein 1


(Homo sapiens (Human))		BDBM50516143
PNG
(CHEMBL4546577)
Show SMILES COc1ccc(NC(=O)C2CCN(CC2)c2ncccc2Cl)cc1Cl
Show InChI InChI=1S/C18H19Cl2N3O2/c1-25-16-5-4-13(11-15(16)20)22-18(24)12-6-9-23(10-7-12)17-14(19)3-2-8-21-17/h2-5,8,11-12H,6-7,9-10H2,1H3,(H,22,24)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 100n/an/an/an/an/an/a



Janssen Research & Development, LLC

Curated by ChEMBL


Assay Description
Inhibition of strep-tagged and His-tagged full length MALT1 protease (1 to 824 residues) (unknown origin) expressed in baculovirus infected insect ce...

Bioorg Med Chem Lett 29: (2019)


Article DOI: 10.1016/j.bmcl.2019.126743
BindingDB Entry DOI: 10.7270/Q2DV1P7R
More data for this
Ligand-Target Pair