Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neutrophil elastase (Homo sapiens (Human)) | BDBM50281013 ((R)-3-Benzyl-6-isopropyl-7-oxo-4-thia-1-aza-bicycl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of Human leukocyte elastase | Bioorg Med Chem Lett 3: 2277-2282 (1993) Article DOI: 10.1016/S0960-894X(01)80939-2 BindingDB Entry DOI: 10.7270/Q2WW7HMK | |||||||||||
More data for this Ligand-Target Pair |