Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nuclear receptor subfamily 1 group I member 2 (Homo sapiens (Human)) | BDBM50510069![]() (CHEMBL4467862) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a |
University of Perugia Curated by ChEMBL | Assay Description Agonist activity at PXR (unknown origin) by AlphaScreen assay | ACS Med Chem Lett 10: 677-681 (2019) Article DOI: 10.1021/acsmedchemlett.8b00459 BindingDB Entry DOI: 10.7270/Q2GT5RHZ | |||||||||||
More data for this Ligand-Target Pair |