Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 (Homo sapiens (Human)) | BDBM50518732![]() (CHEMBL4473488) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 5.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Nagoya Citi University Curated by ChEMBL | Assay Description Irreversible inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition a... | Bioorg Med Chem Lett 29: 353-356 (2019) Article DOI: 10.1016/j.bmcl.2018.12.044 BindingDB Entry DOI: 10.7270/Q27D2ZH0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 (Homo sapiens (Human)) | BDBM50518732![]() (CHEMBL4473488) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Nagoya Citi University Curated by ChEMBL | Assay Description Inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition and measured f... | Bioorg Med Chem Lett 29: 353-356 (2019) Article DOI: 10.1016/j.bmcl.2018.12.044 BindingDB Entry DOI: 10.7270/Q27D2ZH0 | |||||||||||
More data for this Ligand-Target Pair |