Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM50216939 (CHEMBL246207 | {(S)-5-[2-(2-biphenyl-4-yl-5-methyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.72E+3 | n/a | n/a | n/a | n/a |
Bayer Research Center Curated by ChEMBL | Assay Description Agonist activity at PPARalpha by FRET assay | Bioorg Med Chem Lett 17: 4369-73 (2007) Article DOI: 10.1016/j.bmcl.2007.03.057 BindingDB Entry DOI: 10.7270/Q2GX4B8H | |||||||||||
More data for this Ligand-Target Pair |