Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50148092 (7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA) | J Med Chem 47: 3255-63 (2004) Article DOI: 10.1021/jm030621d BindingDB Entry DOI: 10.7270/Q2JW8DB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50148092 (7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 360 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro transcriptional activation by human PPAR gamma Gal4 chimera | J Med Chem 47: 3255-63 (2004) Article DOI: 10.1021/jm030621d BindingDB Entry DOI: 10.7270/Q2JW8DB1 | |||||||||||
More data for this Ligand-Target Pair |