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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50023322'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50023322
PNG
(1-{6-[(2,3-Dimethyl-11-oxo-11H-pyrido[2,1-b]quinaz...)
Show SMILES Cc1cc2nc3ccc(cn3c(=O)c2cc1C)C(=O)NCCCCCC[n+]1ccccc1
Show InChI InChI=1S/C26H28N4O2/c1-19-16-22-23(17-20(19)2)28-24-11-10-21(18-30(24)26(22)32)25(31)27-12-6-3-4-7-13-29-14-8-5-9-15-29/h5,8-11,14-18H,3-4,6-7,12-13H2,1-2H3/p+1
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PubMed
n/an/a>1.00E+3n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

Curated by ChEMBL


Assay Description
Ability to inhibit platelet activating factor (PAF) binding to platelets by 50% was determined by using [3H]-PAF as radioligand

J Med Chem 31: 466-72 (1988)


BindingDB Entry DOI: 10.7270/Q2KK99S6
More data for this
Ligand-Target Pair