Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-derived growth factor receptor alpha/beta (Mus musculus (mouse)) | BDBM50256044![]() (5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...) | MMDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 177 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description Antagonist activity at muscarinic receptor M2 assessed as contraction of electrically-stimulated guinea pig left atria | Citation and Details | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-derived growth factor receptor alpha/beta (Mus musculus (mouse)) | BDBM50256044![]() (5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...) | MMDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description Activity at human B2 receptor transfected in CHO cells assessed as ability to antagonize BK-induced inositol-phosphate accumulation | Citation and Details | |||||||||||
More data for this Ligand-Target Pair |