Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-derived growth factor receptor alpha/beta (Mus musculus (mouse)) | BDBM5931![]() (BMS-387072 | CHEMBL296468 | N-(5-{[(5-tert-butyl-1...) | MMDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description Ability to displace [3H]glycine from strychnine-insensitive glycine receptor | Citation and Details | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-derived growth factor receptor alpha/beta (Mus musculus (mouse)) | BDBM5931![]() (BMS-387072 | CHEMBL296468 | N-(5-{[(5-tert-butyl-1...) | MMDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description Blocking activity against Beta-1 adrenergic receptor in spontaneously beating guinea pig atrial preparations | Citation and Details | |||||||||||
More data for this Ligand-Target Pair |