Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552370![]() (US11312727, Compound 148BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552370![]() (US11312727, Compound 148BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552370![]() (US11312727, Compound 148BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a |
TBA | Assay Description Human lung carcinoma A549 cells (ATCC, Manassas, Va.) were plated at a density of 5×104 cells/mL (10×103 cells/well) in assay media (Ham's F12 me... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552370![]() (US11312727, Compound 148BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Human lung carcinoma A549 cells (ATCC, Manassas, Va.) were plated at a density of 5×104 cells/mL (10×103 cells/well) in assay media (Ham's F12 me... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair |