Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50287520![]() (CHEMBL4159883) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | 2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Displacement of fluorescent-labelled dofetilide from human ERG expressed in HEK293 cell membrane homogenates | ACS Med Chem Lett 9: 125-130 (2018) Article DOI: 10.1021/acsmedchemlett.7b00481 BindingDB Entry DOI: 10.7270/Q2KH0QVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50287520![]() (CHEMBL4159883) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | >4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Displacement of fluorescent-labelled dofetilide from human ERG expressed in HEK293 cell membrane homogenates | ACS Med Chem Lett 9: 125-130 (2018) Article DOI: 10.1021/acsmedchemlett.7b00481 BindingDB Entry DOI: 10.7270/Q2KH0QVZ | |||||||||||
More data for this Ligand-Target Pair |