Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50432396![]() (CHEMBL2348780) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
ReveraGen BioPharma, Inc. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem 21: 2241-9 (2013) Article DOI: 10.1016/j.bmc.2013.02.009 BindingDB Entry DOI: 10.7270/Q2639R3C | |||||||||||
More data for this Ligand-Target Pair |