BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Probable G-protein coupled receptor 34' and Ligand = 'BDBM50238930'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Probable G-protein coupled receptor 34 (Mus musculus)	BDBM50238930 (CHEMBL4094801) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	1.95E+3	n/a	n/a	n/a	n/a
The University of Tokyo Curated by ChEMBL					Assay Description Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...				J Med Chem 60: 6384-6399 (2017) Article DOI: 10.1021/acs.jmedchem.7b00693 BindingDB Entry DOI: 10.7270/Q2FX7CR1
The University of Tokyo Curated by ChEMBL					More data for this Ligand-Target Pair
Probable G-protein coupled receptor 34 (Mus musculus)	BDBM50238930 (CHEMBL4094801) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a
The University of Tokyo Curated by ChEMBL					Assay Description Opioid receptor affinity against Opioid receptor kappa 1 by using the curve-fitting program LIGAND				J Med Chem 60: 6384-6399 (2017) Article DOI: 10.1021/acs.jmedchem.7b00693 BindingDB Entry DOI: 10.7270/Q2FX7CR1
The University of Tokyo Curated by ChEMBL					More data for this Ligand-Target Pair