Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prolyl endopeptidase (Sus scrofa) | BDBM50291163 (4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyr...) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzyme | Bioorg Med Chem Lett 7: 533-538 (1997) Article DOI: 10.1016/S0960-894X(97)00057-7 BindingDB Entry DOI: 10.7270/Q28S4QF2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl endopeptidase (Sus scrofa) | BDBM50291163 (4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyr...) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Meiji Seika Kaisha, Ltd Curated by ChEMBL | Assay Description In vitro inhibitory activity against prolyl endopeptidase (PEP) | J Med Chem 37: 3492-502 (1994) BindingDB Entry DOI: 10.7270/Q2RB73N9 | |||||||||||
More data for this Ligand-Target Pair |