Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteasome subunit beta type-5 (Homo sapiens (Human)) | BDBM50554386 (CHEMBL4758484) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 244 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human constitutive 20S proteasome beta 5 chymotrypsin-like activity | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01520 BindingDB Entry DOI: 10.7270/Q22R3WB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit beta type-5 (Homo sapiens (Human)) | BDBM50554386 (CHEMBL4758484) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human 20S constitutive proteasome beta 5 chymotrypsin-like activity in human HeLa cells incubated for 2 hrs by proteasome-Glo assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01520 BindingDB Entry DOI: 10.7270/Q22R3WB6 | |||||||||||
More data for this Ligand-Target Pair |