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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50583766'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Pyroglutamylated RF-amide peptide receptor


(Homo sapiens (Human))		BDBM50583766
PNG
(CHEMBL5074999)
Show SMILES [#7]-[#6](=[#7])-[#7]-[#6]-[#6]-[#6]-[#6@@H](-[#7]-[#6](=O)\[#6]=[#6](\c1ccccc1)-c1ccccc1)-[#6](=O)-[#7]-[#6@H](-[#6]-c1ccccc1)-[#6](-[#7])=O |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
>5.00E+3n/an/an/an/an/an/an/an/a


TBA

Assay Description
Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting method

Citation and Details

Article DOI: 10.1021/acs.jmedchem.1c00256
BindingDB Entry DOI: 10.7270/Q2VX0MDH
More data for this
Ligand-Target Pair