BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM50316026'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
RAC-alpha serine/threonine-protein kinase (Homo sapiens (Human))	BDBM50316026 ((S)-N-((6S,9S,12S,15S,18S)-1-amino-15-(aminomethyl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	940	n/a	n/a	n/a	n/a	n/a	n/a
The Hebrew University of Jerusalem Curated by ChEMBL					Assay Description Inhibition of Akt using RPRTSSF peptide and [gamma32]ATP by cell-free radioactive assay				J Med Chem 54: 5154-64 (2011) Article DOI: 10.1021/jm2003969 BindingDB Entry DOI: 10.7270/Q26D5TBX
The Hebrew University of Jerusalem Curated by ChEMBL					More data for this Ligand-Target Pair
RAC-alpha serine/threonine-protein kinase (Homo sapiens (Human))	BDBM50316026 ((S)-N-((6S,9S,12S,15S,18S)-1-amino-15-(aminomethyl...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	940	n/a	n/a	n/a	n/a	n/a	n/a
The Hebrew University of Jerusalem Curated by ChEMBL					Assay Description Inhibition of PKB by radioactive kinase assay				Bioorg Med Chem 18: 2976-85 (2010) Article DOI: 10.1016/j.bmc.2010.02.031 BindingDB Entry DOI: 10.7270/Q2KD1Z2W
The Hebrew University of Jerusalem Curated by ChEMBL					More data for this Ligand-Target Pair