Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
RAC-alpha serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50316357 (2-(5-{[(2S)-2-Amino-3-(2-chlorophenyl)propyl]oxy}p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 793 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Inhibition of AKT | Eur J Med Chem 45: 1379-86 (2010) Article DOI: 10.1016/j.ejmech.2009.12.036 BindingDB Entry DOI: 10.7270/Q2HD7VT5 | |||||||||||
More data for this Ligand-Target Pair |