Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50563231 (CHEMBL4780098) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.88E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01533 BindingDB Entry DOI: 10.7270/Q2XW4PHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50563231 (CHEMBL4780098) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.59E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01533 BindingDB Entry DOI: 10.7270/Q2XW4PHG | |||||||||||
More data for this Ligand-Target Pair |