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Found 1 hit Enz. Inhib. hit(s) with Target = 'Reverse transcriptase' and Ligand = 'BDBM50484327'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50484327
PNG
(CHEMBL1835502)
Show SMILES Fc1ccc(OCCn2ccc(=O)[nH]c2=O)c(c1)C(=O)c1ccccc1
Show InChI InChI=1S/C19H15FN2O4/c20-14-6-7-16(15(12-14)18(24)13-4-2-1-3-5-13)26-11-10-22-9-8-17(23)21-19(22)25/h1-9,12H,10-11H2,(H,21,23,25)
PDB
MMDB

UniProtKB/TrEMBL

B.MOAD
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
 2.60E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...

Bioorg Med Chem 19: 5794-802 (2011)


Article DOI: 10.1016/j.bmc.2011.08.025
BindingDB Entry DOI: 10.7270/Q2057JRG
More data for this
Ligand-Target Pair