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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha/beta' and Ligand = 'BDBM573138'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha/beta


(Homo sapiens (Human))
BDBM573138
PNG
(US11453673, Example 4)
Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1CCC1)C1(CC1)C1CC1
PDB

UniProtKB/SwissProt

antibodypedia
antibodypedia
GoogleScholar
AffyNet 
Purchase

MCE
PC cid
PC sid
UniChem
US Patent
n/an/a>1.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Table 7: The following phosphodiesterase activities are measured using [3H]cGMP as reaction substrate: human PDE6A/6B. The catalytic active form of h...


Citation and Details

BindingDB Entry DOI: 10.7270/Q22Z18RF
More data for this
Ligand-Target Pair