Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Serine/threonine-protein kinase ULK1 (Homo sapiens (Human)) | BDBM50271371 (CHEMBL4125718) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
Sichuan Universitt China Hospital Curated by ChEMBL | Assay Description Activation of recombinant human N-terminal GST-tagged ULK1 (1 to 649 residues) expressed in baculovirus infected Sf9 cells using MBP as substrate aft... | J Med Chem 61: 6491-6500 (2018) Article DOI: 10.1021/acs.jmedchem.7b01684 BindingDB Entry DOI: 10.7270/Q2DN47KX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase ULK1 (Homo sapiens (Human)) | BDBM50271371 (CHEMBL4125718) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a | |
TBA | Assay Description Antagonist potency against histamine H3 receptor in an electrically stimulated guinea pig ileum | Citation and Details | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase ULK1 (Homo sapiens (Human)) | BDBM50271371 (CHEMBL4125718) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01291 BindingDB Entry DOI: 10.7270/Q24J0K63 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase ULK1 (Homo sapiens (Human)) | BDBM50271371 (CHEMBL4125718) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
China Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of ULK1 (unknown origin) using MBP as substrate after 60 mins by ADP-Glo assay | J Med Chem 61: 4656-4687 (2018) Article DOI: 10.1021/acs.jmedchem.7b01019 BindingDB Entry DOI: 10.7270/Q2RR22GW | |||||||||||
More data for this Ligand-Target Pair |