Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human)) | BDBM50509368![]() (CHEMBL4475097) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
UiT - The Arctic University of Norway Curated by ChEMBL | Assay Description Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assay | J Med Chem 62: 10167-10181 (2019) Article DOI: 10.1021/acs.jmedchem.9b01006 BindingDB Entry DOI: 10.7270/Q26M3B4R | |||||||||||
More data for this Ligand-Target Pair |