Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein phosphatase 2A activator (Homo sapiens (Human)) | BDBM40785![]() (Calyculinamide A (18)) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo | Assay Description Protein phosphatase inhibitory activity of calyculin derivatives. | Chem Biol 9: 309-19 (2002) Article DOI: 10.1016/S1074-5521(02)00118-7 BindingDB Entry DOI: 10.7270/Q2W66J5W | |||||||||||
More data for this Ligand-Target Pair |