Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50041113![]() (2-(3-Methoxy-phenyl)-1H-quinolin-4-one | CHEMBL276...) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of bovine brain tubulin polymerization (ITP). | J Med Chem 41: 1155-62 (1998) Article DOI: 10.1021/jm9707479 BindingDB Entry DOI: 10.7270/Q2RN3BKW | |||||||||||
More data for this Ligand-Target Pair |