Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent dopamine transporter (Homo sapiens (Human)) | BDBM50459625 (CHEMBL4205254) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Organix Inc Curated by ChEMBL | Assay Description Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranes | J Med Chem 61: 9121-9131 (2018) Article DOI: 10.1021/acs.jmedchem.8b00542 BindingDB Entry DOI: 10.7270/Q2KH0QZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Homo sapiens (Human)) | BDBM50459625 (CHEMBL4205254) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Organix Inc Curated by ChEMBL | Assay Description Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranes | J Med Chem 61: 9121-9131 (2018) Article DOI: 10.1021/acs.jmedchem.8b00542 BindingDB Entry DOI: 10.7270/Q2KH0QZ9 | |||||||||||
More data for this Ligand-Target Pair |