Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent phosphate transport protein 2A (Homo sapiens) | BDBM50341383 (CHEMBL4175607) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 750 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Displacement of (C[3H]3) from NaPi2a (unknown origin) expressed in HEK293 cell membranes coexpressing tetracyclin after 1 hr by scintillation countin... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transport protein 2A (Homo sapiens) | BDBM50341383 (CHEMBL4175607) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of human NaPi2a expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transport protein 2A (Rattus norvegicus) | BDBM50341383 (CHEMBL4175607) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of rat NaPi2a expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20 t... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent phosphate transport protein 2A (Mus musculus) | BDBM50341383 (CHEMBL4175607) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of mouse NaPi2a expressed in HEK293 cells coexpressing tetracyclin assessed as reduction in uptake of 33P-radiolabeled Pi incubated for 20... | ACS Med Chem Lett 9: 440-445 (2018) Article DOI: 10.1021/acsmedchemlett.8b00013 BindingDB Entry DOI: 10.7270/Q26T0Q7K | |||||||||||
More data for this Ligand-Target Pair |