Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent serotonin transporter (Rattus norvegicus (rat)) | BDBM50057136 ((2-Benzo[b]thiophen-5-yl-ethyl)-((R)-5-methoxy-1,2...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 52.8 | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Park Curated by ChEMBL | Assay Description Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortex | J Med Chem 40: 1049-62 (1997) Article DOI: 10.1021/jm960723m BindingDB Entry DOI: 10.7270/Q2CF9P6W | |||||||||||
More data for this Ligand-Target Pair |