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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Solute carrier family 2, facilitated glucose transporter member 4' and Ligand = 'BDBM50565143'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Solute carrier family 2, facilitated glucose transporter member 4


(Homo sapiens)
BDBM50565143
PNG
(CHEMBL4793560)
Show SMILES O=C(CN1C(=O)S\C(=C\c2ccco2)C1=O)Nc1nc2ccccc2s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
Purchase

MCE
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 6.80E+3n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112603
BindingDB Entry DOI: 10.7270/Q25Q50T2
More data for this
Ligand-Target Pair