Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sterol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50284875 (CHEMBL41967 | Phosphoric acid mono-(4-{(4R,5R)-2-[...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 2.55E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibitory activity against acylcoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit thoracic aorta | Bioorg Med Chem Lett 5: 1581-1586 (1995) Article DOI: 10.1016/0960-894X(95)00275-X BindingDB Entry DOI: 10.7270/Q2222TPK | |||||||||||
More data for this Ligand-Target Pair |