Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sucrase-isomaltase, intestinal (Rattus norvegicus (Rat)) | BDBM50333456 ((2S,3S,4S,5S)-2-(hydroxymethyl)-5-pentylpyrrolidin...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
Tohoku Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of Wistar rat small intestine sucrase after 30 mins | Bioorg Med Chem Lett 21: 738-41 (2011) Article DOI: 10.1016/j.bmcl.2010.11.112 BindingDB Entry DOI: 10.7270/Q2D21XVS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sucrase-isomaltase, intestinal (Rattus norvegicus (Rat)) | BDBM50333456 ((2S,3S,4S,5S)-2-(hydroxymethyl)-5-pentylpyrrolidin...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Toyama Curated by ChEMBL | Assay Description Inhibition of rat intestinal sucrase using sucrose as substrate | J Med Chem 55: 10347-62 (2012) Article DOI: 10.1021/jm301304e BindingDB Entry DOI: 10.7270/Q2K35VTX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sucrase-isomaltase, intestinal (Rattus norvegicus (Rat)) | BDBM50333456 ((2S,3S,4S,5S)-2-(hydroxymethyl)-5-pentylpyrrolidin...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Toyama Curated by ChEMBL | Assay Description Inhibition of rat intestinal isomaltase using isomoltose as substrate | J Med Chem 55: 10347-62 (2012) Article DOI: 10.1021/jm301304e BindingDB Entry DOI: 10.7270/Q2K35VTX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sucrase-isomaltase, intestinal (Rattus norvegicus (Rat)) | BDBM50333456 ((2S,3S,4S,5S)-2-(hydroxymethyl)-5-pentylpyrrolidin...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tohoku Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of Wistar rat small intestine isomaltase after 30 mins | Bioorg Med Chem Lett 21: 738-41 (2011) Article DOI: 10.1016/j.bmcl.2010.11.112 BindingDB Entry DOI: 10.7270/Q2D21XVS | |||||||||||
More data for this Ligand-Target Pair |