Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Taste receptor type 1 member 1/3 (Homo sapiens (Human)) | BDBM525952 (US11185100, TABLE 6.5) | UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a |
TBA | Assay Description HEK293 cells that stably express T1R3 and inducibly express T1R1 were exposed to nucleotide derivatives alone to activate the umami receptor. Activat... | Citation and Details BindingDB Entry DOI: 10.7270/Q2KP859X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Taste receptor type 1 member 1/3 (Homo sapiens (Human)) | BDBM525952 (US11185100, TABLE 6.5) | UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a |
TBA | Assay Description The concentration of alanine is 20 mM, and the concentration of IMP is 0.2 mM. | Citation and Details BindingDB Entry DOI: 10.7270/Q2KP859X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Taste receptor type 1 member 1/3 (Homo sapiens (Human)) | BDBM525952 (US11185100, TABLE 6.5) | UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 7.20E+5 | n/a | n/a | n/a | n/a |
TBA | Assay Description The concentration of IMP is 0.2 mM. | Citation and Details BindingDB Entry DOI: 10.7270/Q2KP859X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Taste receptor type 1 member 1/3 (Homo sapiens (Human)) | BDBM525952 (US11185100, TABLE 6.5) | UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a |
TBA | Assay Description The concentration of alanine is 20 mM. | Citation and Details BindingDB Entry DOI: 10.7270/Q2KP859X | |||||||||||
More data for this Ligand-Target Pair |