Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM151746'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human))	BDBM151746 (US8987445, 182) Show SMILES Cc1cc2ccccc2nc1N(Cc1ccc(cc1)C(F)(F)C1CC1)S(=O)(=O)c1ccc(cc1)C(O)=O Show InChI InChI=1S/C28H24F2N2O4S/c1-18-16-21-4-2-3-5-25(21)31-26(18)32(37(35,36)24-14-8-20(9-15-24)27(33)34)17-19-6-10-22(11-7-19)28(29,30)23-12-13-23/h2-11,14-16,23H,12-13,17H2,1H3,(H,33,34)	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	37
Mitsubishi Tanabe Pharma Corporation US Patent					Assay Description The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+ sensitive fluorescent dy...				US Patent US8987445 (2015) BindingDB Entry DOI: 10.7270/Q2BZ64R5
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