Compile Data Set for Download or QSAR

Found 2 hits Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50317560'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily M member 8 (Rattus norvegicus (Rat))	BDBM50317560 (CHEMBL1095102 | N-[(1R,2S,5R)-2-Isopropyl-5-methyl...) Show SMILES CC(C)[C@@H]1CC[C@@H](C)C[C@H]1NC(=O)CCCCCCCc1ccccc1 |r| Show InChI InChI=1S/C24H39NO/c1-19(2)22-17-16-20(3)18-23(22)25-24(26)15-11-6-4-5-8-12-21-13-9-7-10-14-21/h7,9-10,13-14,19-20,22-23H,4-6,8,11-12,15-18H2,1-3H3,(H,25,26)/t20-,22+,23-/m1/s1	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
Sapienza Universit£ di Roma Curated by ChEMBL					Assay Description Antagonist activity at rat TRMP8 receptor expressed in HEK293 cells assessed as menthol-induced calcium elevation				Bioorg Med Chem Lett 20: 2729-32 (2010) Article DOI: 10.1016/j.bmcl.2010.03.076 BindingDB Entry DOI: 10.7270/Q27M083N
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Rattus norvegicus (Rat))	BDBM50317560 (CHEMBL1095102 | N-[(1R,2S,5R)-2-Isopropyl-5-methyl...) Show SMILES CC(C)[C@@H]1CC[C@@H](C)C[C@H]1NC(=O)CCCCCCCc1ccccc1 |r| Show InChI InChI=1S/C24H39NO/c1-19(2)22-17-16-20(3)18-23(22)25-24(26)15-11-6-4-5-8-12-21-13-9-7-10-14-21/h7,9-10,13-14,19-20,22-23H,4-6,8,11-12,15-18H2,1-3H3,(H,25,26)/t20-,22+,23-/m1/s1	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
Sapienza Universit£ di Roma Curated by ChEMBL					Assay Description Antagonist activity at rat TRMP8 receptor expressed in HEK293 cells assessed as menthol-induced calcium elevation				Bioorg Med Chem Lett 20: 2729-32 (2010) Article DOI: 10.1016/j.bmcl.2010.03.076 BindingDB Entry DOI: 10.7270/Q27M083N
					More data for this Ligand-Target Pair