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Compile Data Set for Download or QSAR

Found 2 hits Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 4' and Ligand = 'BDBM539876'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Transient receptor potential cation channel subfamily V member 4


(Homo sapiens (Human))
BDBM539876
PNG
(2-chloro-4-(difluoro- methyl)benzene-1- sulfonyl c...)
Show SMILES FC(F)c1ccc(c(Cl)c1)S(Cl)(=O)=O
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 5n/an/an/an/an/an/a


TBA

Assay Description
TRPV4 channel activation results in an influx of divalent and monovalent cations including calcium. The resulting changes in intracellular calcium we...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2B85C9Z
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 4


(Homo sapiens (Human))
BDBM539876
PNG
(2-chloro-4-(difluoro- methyl)benzene-1- sulfonyl c...)
Show SMILES FC(F)c1ccc(c(Cl)c1)S(Cl)(=O)=O
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 55n/an/an/an/an/an/a


TBA

Assay Description
TRPV4 channel activation results in an influx of divalent and monovalent cations including calcium. The resulting changes in intracellular calcium we...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2B85C9Z
More data for this
Ligand-Target Pair