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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Type-2 angiotensin II receptor' and Ligand = 'BDBM50284443'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Type-2 angiotensin II receptor


(RAT)		BDBM50284443
PNG
(CHEMBL280456 | [4-(2-Ethyl-6,8-dimethyl-imidazo[1,...)
Show SMILES CCc1nc2c(C)cc(C)nn2c1Cc1ccc(OC(C(O)=O)c2ccccc2)cc1
Show InChI InChI=1S/C25H25N3O3/c1-4-21-22(28-24(26-21)16(2)14-17(3)27-28)15-18-10-12-20(13-11-18)31-23(25(29)30)19-8-6-5-7-9-19/h5-14,23H,4,15H2,1-3H3,(H,29,30)
PDB

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UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
Article
n/an/a 3.00E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for its ability to displace the specific binding ligand [125I]-Sar 1,lle8-AlI from rat midbrain membrane (AT2 receptor)

Bioorg Med Chem Lett 5: 1151-1154 (1995)


Article DOI: 10.1016/0960-894X(95)00185-V
BindingDB Entry DOI: 10.7270/Q2J67GV9
More data for this
Ligand-Target Pair